An Efficient, One-Pot Transamidation of 8-Aminoquinoline Amides Activated by Tertiary-Butyloxycarbonyl
The efficient, one-pot access to the transamidation Postnatal Body of 8-aminoquinoline (8-AQ), notorious for its harsh removal conditions, has been widely employed as an auxiliary in C–H functionalization reactions due to its strong directing ability.In this study, the facile and mild Boc protection of the corresponding 8-AQ Teethers amide wa